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Compound
PGDB_C009246
2 activity records1 related patents
2D structure
CC(C)(O)c1cccn(-c2ccc(-c3cccc(C4CCC(=O)NC4=O)c3Cl)s2)c1=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 97 | % | Concentration series: 1000 nM, 250 nM, 62.5 nM, 15.6 nM, 3.9 nM, 0.98 nM, 0.24 nM, 0 nM | 24 h | VAV1 | - | Jurkat | WO2026041143A1 | PGDB_A040912 | PGDB_C009246 | PGDB_AS000206 | View |
| DC50 | - | <= | 10 | nM | - | — | VAV1 | - | Jurkat | WO2026041143A1 | PGDB_A061325 | PGDB_C009246 | PGDB_AS001882 | View |