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C=CC(=O)N1CCC(F)(F)CC1c1cc2cc(-c3ccccc3O)nnc2[nH]1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | < | 30 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A007634 | PGDB_C010281 | PGDB_AS002120 | View | |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A009442 | PGDB_C010281 | PGDB_AS000431 | View | |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A021416 | PGDB_C010281 | PGDB_AS002120 | View | |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A024709 | PGDB_C010281 | PGDB_AS001961 | View | |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A033839 | PGDB_C010281 | PGDB_AS000431 | View | |
| DC50 | - | < | 0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A042321 | PGDB_C010281 | PGDB_AS000900 | View | |
| DC50 | - | < | 0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A046127 | PGDB_C010281 | PGDB_AS000900 | View | |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A059170 | PGDB_C010281 | PGDB_AS001961 | View |