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SIMM · NJU
Assay
PGDB_AS000431
System: cell_based
Target: SMARCA4
Cell line: HeLa
Assay context summary
Assay context
643 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
SMARCA4
E3
Not specified
Cell line
HeLa
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
643 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007044
PGDB_C010699
PGDB_AS000431
View
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007076
PGDB_C010669
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007175
PGDB_C010563
PGDB_AS000431
View
DC50
-
>
5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007224
PGDB_C010360
PGDB_AS000431
View
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007250
PGDB_C010463
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007398
PGDB_C010452
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007540
PGDB_C010530
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007623
PGDB_C010229
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007689
PGDB_C010510
PGDB_AS000431
View
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007756
PGDB_C010481
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A007995
PGDB_C010430
PGDB_AS000431
View
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A008044
PGDB_C010225
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A008656
PGDB_C010447
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A008750
PGDB_C010255
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A008784
PGDB_C010238
PGDB_AS000431
View
DC50
-
>
5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A008867
PGDB_C010841
PGDB_AS000431
View
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A008936
PGDB_C010576
PGDB_AS000431
View
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A009047
PGDB_C010836
PGDB_AS000431
View
DC50
-
<
0.5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A009056
PGDB_C010783
PGDB_AS000431
View
DC50
-
=
0.5-5
uM
-
—
SMARCA4
-
HeLa
WO2025101944
PGDB_A009240
PGDB_C010468
PGDB_AS000431
View