Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C010468
8 activity records1 related patents
2D structure
C=CC(=O)N1CC[C@@H](F)C(c2cc3cc(-c4ccccc4O)nnc3[nH]2)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A009240 | PGDB_C010468 | PGDB_AS000431 | View |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A011622 | PGDB_C010468 | PGDB_AS001961 | View |
| % Degradation | - | < | 30 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A048956 | PGDB_C010468 | PGDB_AS002120 | View |
| DC50 | - | < | 0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A049020 | PGDB_C010468 | PGDB_AS000900 | View |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A063107 | PGDB_C010468 | PGDB_AS001961 | View |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A066601 | PGDB_C010468 | PGDB_AS000431 | View |
| DC50 | - | < | 0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A067037 | PGDB_C010468 | PGDB_AS000900 | View |
| % Degradation | - | < | 30 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A068420 | PGDB_C010468 | PGDB_AS002120 | View |