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C=CC(=O)N1CC2(CCCC2c2[nH]c3nnc(-c4cccc(F)c4O)cc3c2C)C1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | < | 0.5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A007044 | PGDB_C010699 | PGDB_AS000431 | View | |
| % Degradation | - | > | 70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A014404 | PGDB_C010699 | PGDB_AS001961 | View | |
| % Degradation | - | > | 70 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A016850 | PGDB_C010699 | PGDB_AS002120 | View | |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A025857 | PGDB_C010699 | PGDB_AS002120 | View | |
| % Degradation | - | > | 70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A052563 | PGDB_C010699 | PGDB_AS001961 | View | |
| DC50 | - | < | 0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A062424 | PGDB_C010699 | PGDB_AS000900 | View | |
| DC50 | - | < | 0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A074146 | PGDB_C010699 | PGDB_AS000900 | View | |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A074614 | PGDB_C010699 | PGDB_AS000431 | View |