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C=CC(=O)N1CC[C@@H](c2[nH]c3nnc(-c4ccccc4O)cc3c2[C@H]2COC[C@@H]2F)C1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | < | 0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A007184 | PGDB_C010778 | PGDB_AS000900 | View | |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A029705 | PGDB_C010778 | PGDB_AS000431 | View | |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A041128 | PGDB_C010778 | PGDB_AS002120 | View | |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A043920 | PGDB_C010778 | PGDB_AS000900 | View | |
| % Degradation | - | > | 70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A048163 | PGDB_C010778 | PGDB_AS001961 | View | |
| % Degradation | - | < | 30 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A048183 | PGDB_C010778 | PGDB_AS002120 | View | |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2025101944 | PGDB_A050203 | PGDB_C010778 | PGDB_AS000431 | View | |
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2025101944 | PGDB_A069926 | PGDB_C010778 | PGDB_AS001961 | View |