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Compound
PGDB_C010912
4 activity records1 related patents
2D structure
Fc1ccc2nc(CNc3cc(N4CC5CCC(C4)O5)nn4c(C(F)(F)F)cnc34)[nH]c2c1FCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 0.1 | uM | - | — | CDK12 | - | - | WO2025110815A1 | PGDB_A011164 | PGDB_C010912 | PGDB_AS002095 | View |
| IC50 | - | <= | 0.3 | uM | - | — | POLR2A | - | - | WO2025110815A1 | PGDB_A037131 | PGDB_C010912 | PGDB_AS000589 | View |
| IC50 | - | <= | 0.1 | uM | - | — | CDK13 | - | - | WO2025110815A1 | PGDB_A043092 | PGDB_C010912 | PGDB_AS001146 | View |
| IC50 | - | <= | 0.05 | uM | - | — | - | - | MDA-MB-231 | WO2025110815A1 | PGDB_A056464 | PGDB_C010912 | PGDB_AS000344 | View |