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CN1CCN(c2cc(NCc3nc4cc(Cl)c(Cl)cc4[nH]3)c3ncc(C(F)(F)F)n3n2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 0.2 | uM | - | — | - | - | AGS | WO2025110815A1 | PGDB_A011938 | PGDB_C010932 | PGDB_AS000697 | View | |
| IC50 | - | <= | 0.2 | uM | - | — | - | - | MKN45 | WO2025110815A1 | PGDB_A013164 | PGDB_C010932 | PGDB_AS000058 | View | |
| IC50 | - | <= | 0.2 | uM | - | — | - | - | KATO-III | WO2025110815A1 | PGDB_A017067 | PGDB_C010932 | PGDB_AS001821 | View | |
| IC50 | - | <= | 0.05 | uM | - | — | - | - | HCC70 | WO2025110815A1 | PGDB_A041867 | PGDB_C010932 | PGDB_AS001231 | View | |
| IC50 | - | <= | 0.05 | uM | - | — | - | - | MDA-MB-231 | WO2025110815A1 | PGDB_A046135 | PGDB_C010932 | PGDB_AS000344 | View | |
| IC50 | - | <= | 0.1 | uM | - | — | CDK13 | - | - | WO2025110815A1 | PGDB_A055799 | PGDB_C010932 | PGDB_AS001146 | View | |
| IC50 | - | <= | 0.2 | uM | - | — | - | - | SNU-1 | WO2025110815A1 | PGDB_A058774 | PGDB_C010932 | PGDB_AS001364 | View | |
| IC50 | - | <= | 0.05 | uM | - | — | - | - | MDA-MB-436 | WO2025110815A1 | PGDB_A060049 | PGDB_C010932 | PGDB_AS002448 | View | |
| IC50 | - | <= | 0.1 | uM | - | — | CDK12 | - | - | WO2025110815A1 | PGDB_A064380 | PGDB_C010932 | PGDB_AS002095 | View | |
| IC50 | - | <= | 0.3 | uM | - | — | POLR2A | - | - | WO2025110815A1 | PGDB_A075280 | PGDB_C010932 | PGDB_AS000589 | View | |
| IC50 | - | <= | 0.05 | uM | - | — | - | - | BT-20 | WO2025110815A1 | PGDB_A077277 | PGDB_C010932 | PGDB_AS000821 | View |