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N[C@H]1CCN(c2cc(NCc3nc4ccc(F)c(F)c4[nH]3)c3ncc(C(F)(F)F)n3n2)C1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 0.1 | uM | - | — | CDK12 | - | - | WO2025110815A1 | PGDB_A007735 | PGDB_C010941 | PGDB_AS002095 | View | |
| IC50 | - | <= | 0.05 | uM | - | — | - | - | MDA-MB-231 | WO2025110815A1 | PGDB_A061843 | PGDB_C010941 | PGDB_AS000344 | View | |
| IC50 | - | <= | 0.1 | uM | - | — | CDK13 | - | - | WO2025110815A1 | PGDB_A069908 | PGDB_C010941 | PGDB_AS001146 | View | |
| IC50 | - | <= | 0.3 | uM | - | — | POLR2A | - | - | WO2025110815A1 | PGDB_A071457 | PGDB_C010941 | PGDB_AS000589 | View |