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Compound
PGDB_C010943
8 activity records1 related patents
2D structure
Nc1ncc(-c2cc(NCc3nc4cc(Cl)c(Cl)cc4[nH]3)c3ncc(C(F)(F)F)n3n2)cn1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 0.2 | uM | - | — | - | - | MKN1 | WO2025110815A1 | PGDB_A008972 | PGDB_C010943 | PGDB_AS000785 | View |
| IC50 | - | <= | 0.05 | uM | - | — | - | - | MDA-MB-231 | WO2025110815A1 | PGDB_A033444 | PGDB_C010943 | PGDB_AS000344 | View |
| IC50 | - | <= | 0.3 | uM | - | — | POLR2A | - | - | WO2025110815A1 | PGDB_A036265 | PGDB_C010943 | PGDB_AS000589 | View |
| IC50 | - | <= | 0.2 | uM | - | — | - | - | SW480 | WO2025110815A1 | PGDB_A042739 | PGDB_C010943 | PGDB_AS002136 | View |
| IC50 | - | <= | 0.1 | uM | - | — | CDK12 | - | - | WO2025110815A1 | PGDB_A043864 | PGDB_C010943 | PGDB_AS002095 | View |
| IC50 | - | <= | 0.2 | uM | - | — | - | - | HCT15 | WO2025110815A1 | PGDB_A044429 | PGDB_C010943 | PGDB_AS001666 | View |
| IC50 | - | <= | 0.1 | uM | - | — | CDK13 | - | - | WO2025110815A1 | PGDB_A052166 | PGDB_C010943 | PGDB_AS001146 | View |
| IC50 | - | <= | 0.2 | uM | - | — | - | - | AGS | WO2025110815A1 | PGDB_A056187 | PGDB_C010943 | PGDB_AS000706 | View |