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FC(F)(F)c1cnc2c(NCc3cc4ncccc4[nH]3)cc(N3CCOCC3)nn12| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 0.1 | uM | - | — | CDK13 | - | - | WO2025110815A1 | PGDB_A010183 | PGDB_C010970 | PGDB_AS001146 | View | |
| IC50 | - | <= | 0.1 | uM | - | — | CDK12 | - | - | WO2025110815A1 | PGDB_A023476 | PGDB_C010970 | PGDB_AS002095 | View | |
| IC50 | - | = | 0.3-3 | uM | - | — | POLR2A | - | - | WO2025110815A1 | PGDB_A033527 | PGDB_C010970 | PGDB_AS000589 | View | |
| IC50 | - | = | 0.05-0.5 | uM | - | — | - | - | MDA-MB-231 | WO2025110815A1 | PGDB_A037520 | PGDB_C010970 | PGDB_AS000344 | View |