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Compound
PGDB_C010974
4 activity records1 related patents
2D structure
NC(=O)N1CCN(c2cc(NCc3nc4ccc(F)c(F)c4[nH]3)c3ncc(C(F)(F)F)n3n2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.3-3 | uM | - | — | POLR2A | - | - | WO2025110815A1 | PGDB_A010663 | PGDB_C010974 | PGDB_AS000589 | View |
| IC50 | - | = | 0.05-0.5 | uM | - | — | - | - | MDA-MB-231 | WO2025110815A1 | PGDB_A028904 | PGDB_C010974 | PGDB_AS000344 | View |
| IC50 | - | <= | 0.1 | uM | - | — | CDK13 | - | - | WO2025110815A1 | PGDB_A040524 | PGDB_C010974 | PGDB_AS001146 | View |
| IC50 | - | <= | 0.1 | uM | - | — | CDK12 | - | - | WO2025110815A1 | PGDB_A077510 | PGDB_C010974 | PGDB_AS002095 | View |