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C#Cc1cnc([C@H](C)OC)c(-c2c3c4cc(ccc4n2CC(F)(F)F)-c2csc(n2)C[C@H](NC(=O)[C@H](C(C)C)N2CC[C@]4(CCN(C(=O)[C@H]5[C@@H](C6CC6)N5C)C4)C2)C(=O)N2N[C@H](C(=O)OCC(C)(C)C3)C3CC2C3)c1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1-10 | nM | - | — | KRAS | - | AGS | WO2025214350A1 | PGDB_A017785 | PGDB_C011635 | PGDB_AS000218 | View | |
| IC50 | - | = | 1-10 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A036414 | PGDB_C011635 | PGDB_AS002124 | View | |
| IC50 | - | = | 1-10 | nM | - | — | - | - | AsPC-1 | WO2025214350A1 | PGDB_A042958 | PGDB_C011635 | PGDB_AS001410 | View |