Assay context summary

Assay context

77 activity records
Activity compounds and values

Activity records

77 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C011618
IC50-=100-1000nM-KRAS-AGSWO2025214350A1PGDB_A007012PGDB_C011618PGDB_AS000218View
2D structure for PGDB_C011675
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A009159PGDB_C011675PGDB_AS000218View
2D structure for PGDB_C011647
IC50-=10-100nM-KRAS-AGSWO2025214350A1PGDB_A010197PGDB_C011647PGDB_AS000218View
2D structure for PGDB_C011655
IC50-=10-100nM-KRAS-AGSWO2025214350A1PGDB_A010227PGDB_C011655PGDB_AS000218View
2D structure for PGDB_C011652
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A010819PGDB_C011652PGDB_AS000218View
2D structure for PGDB_C011640
IC50-=10-100nM-KRAS-AGSWO2025214350A1PGDB_A011693PGDB_C011640PGDB_AS000218View
2D structure for PGDB_C011615
IC50-=10-100nM-KRAS-AGSWO2025214350A1PGDB_A012295PGDB_C011615PGDB_AS000218View
2D structure for PGDB_C011601
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A013252PGDB_C011601PGDB_AS000218View
2D structure for PGDB_C011677
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A013286PGDB_C011677PGDB_AS000218View
2D structure for PGDB_C028536
IC50-=10-100nM-KRAS-AGSWO2025214350A1PGDB_A014064PGDB_C028536PGDB_AS000218View
2D structure for PGDB_C011598
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A014912PGDB_C011598PGDB_AS000218View
2D structure for PGDB_C011595
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A015075PGDB_C011595PGDB_AS000218View
2D structure for PGDB_C011656
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A015187PGDB_C011656PGDB_AS000218View
2D structure for PGDB_C011676
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A016354PGDB_C011676PGDB_AS000218View
2D structure for PGDB_C011602
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A016470PGDB_C011602PGDB_AS000218View
2D structure for PGDB_C011590
IC50-=10-100nM-KRAS-AGSWO2025214350A1PGDB_A016740PGDB_C011590PGDB_AS000218View
2D structure for PGDB_C011645
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A017541PGDB_C011645PGDB_AS000218View
2D structure for PGDB_C011635
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A017785PGDB_C011635PGDB_AS000218View
2D structure for PGDB_C011596
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A020410PGDB_C011596PGDB_AS000218View
2D structure for PGDB_C011623
IC50-=1-10nM-KRAS-AGSWO2025214350A1PGDB_A020743PGDB_C011623PGDB_AS000218View