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CO[C@@H](C)c1ncc(C#CCN2CCOCC2)cc1-c1c2c3cc(ccc3n1CC(F)(F)F)N1CCO[C@@H](C[C@H](NC(=O)[C@H](C(C)C)C3CC[C@]4(CCN(C(=O)[C@H]5[C@@H](C6CC6)N5C)C4)C3)C(=O)N3CCC[C@H](N3)C(=O)OCC(C)(C)C2)C1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1-10 | nM | - | — | - | - | AsPC-1 | WO2025214350A1 | PGDB_A010899 | PGDB_C011670 | PGDB_AS001410 | View | |
| IC50 | - | = | 1-10 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A031809 | PGDB_C011670 | PGDB_AS002124 | View | |
| IC50 | - | = | 1-10 | nM | - | — | KRAS | - | AGS | WO2025214350A1 | PGDB_A076825 | PGDB_C011670 | PGDB_AS000218 | View |