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Compound
PGDB_C011676
3 activity records1 related patents
2D structure
CCn1c(C2C=C(C#Cc3cncnc3)C=NC2C(C)OC)c2c3cc(ccc31)N1CCO[C@@H](C[C@H](NC(=O)CN3CC[C@]4(CCN(C(=O)[C@@H]5C(C)[C@@H]5C5CC5)C4)C3)C(=O)N3CCC[C@H](N3)C(=O)OCC(C)(C)C2)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1-10 | nM | - | — | KRAS | - | AGS | WO2025214350A1 | PGDB_A016354 | PGDB_C011676 | PGDB_AS000218 | View |
| IC50 | - | = | 1-10 | nM | - | — | - | - | AsPC-1 | WO2025214350A1 | PGDB_A039855 | PGDB_C011676 | PGDB_AS001410 | View |
| IC50 | - | = | 10-100 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A067308 | PGDB_C011676 | PGDB_AS002124 | View |