Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C012056
4 activity records1 related patents
2D structure
C[C@H]1CN(Cc2ccc3onc(N4CCC(=O)NC4=O)c3c2)CCN1CC1CCN(c2ccc(C#N)cn2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 92.2 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A009686 | PGDB_C012056 | PGDB_AS002062 | View |
| Dmax | - | = | 92.2 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A023856 | PGDB_C012056 | PGDB_AS002062 | View |
| DC50 | - | = | 109 | nM | - | — | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A047356 | PGDB_C012056 | PGDB_AS000508 | View |
| DC50 | - | = | 109 | nM | - | — | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A071974 | PGDB_C012056 | PGDB_AS000508 | View |