Assay
PGDB_AS002062
System: cell_basedTarget: WIZ | GSPT1Cell line: HT-1080
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 88.5 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A007840 | PGDB_C012144 | PGDB_AS002062 | View | |
| Dmax | - | = | 92.4 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A007904 | PGDB_C012093 | PGDB_AS002062 | View | |
| Dmax | - | = | 88.9 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A008226 | PGDB_C012053 | PGDB_AS002062 | View | |
| Dmax | - | = | 90.9 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A008761 | PGDB_C012074 | PGDB_AS002062 | View | |
| Dmax | - | = | 93.5 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A008834 | PGDB_C012127 | PGDB_AS002062 | View | |
| Dmax | - | = | 81.2 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A009524 | PGDB_C012067 | PGDB_AS002062 | View | |
| Dmax | - | = | 92.2 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A009686 | PGDB_C012056 | PGDB_AS002062 | View | |
| Dmax | - | = | 87.7 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A010135 | PGDB_C012141 | PGDB_AS002062 | View | |
| Dmax | - | = | 91.3 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A010284 | PGDB_C012077 | PGDB_AS002062 | View | |
| Dmax | - | = | 89.1 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A010328 | PGDB_C012159 | PGDB_AS002062 | View | |
| Dmax | - | = | 92 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A010751 | PGDB_C012110 | PGDB_AS002062 | View | |
| Dmax | - | = | 92.9 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A011068 | PGDB_C012116 | PGDB_AS002062 | View | |
| Dmax | - | = | 79.5 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A011238 | PGDB_C012073 | PGDB_AS002062 | View | |
| Dmax | - | = | 93.3 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A011443 | PGDB_C012099 | PGDB_AS002062 | View | |
| Dmax | - | = | 89.6 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A012171 | PGDB_C012146 | PGDB_AS002062 | View | |
| Dmax | - | = | 87.5 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A012293 | PGDB_C012083 | PGDB_AS002062 | View | |
| Dmax | - | = | 90.5 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A012741 | PGDB_C012121 | PGDB_AS002062 | View | |
| Dmax | - | = | 92.3 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A012841 | PGDB_C012094 | PGDB_AS002062 | View | |
| Dmax | - | = | 95 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A013339 | PGDB_C012088 | PGDB_AS002062 | View | |
| Dmax | - | = | 79.9 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A013770 | PGDB_C012060 | PGDB_AS002062 | View |