Assay context summary

Assay context

116 activity records
Activity compounds and values

Activity records

116 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C012144
Dmax-=88.5%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A007840PGDB_C012144PGDB_AS002062View
2D structure for PGDB_C012093
Dmax-=92.4%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A007904PGDB_C012093PGDB_AS002062View
2D structure for PGDB_C012053
Dmax-=88.9%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A008226PGDB_C012053PGDB_AS002062View
2D structure for PGDB_C012074
Dmax-=90.9%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A008761PGDB_C012074PGDB_AS002062View
2D structure for PGDB_C012127
Dmax-=93.5%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A008834PGDB_C012127PGDB_AS002062View
2D structure for PGDB_C012067
Dmax-=81.2%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A009524PGDB_C012067PGDB_AS002062View
2D structure for PGDB_C012056
Dmax-=92.2%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A009686PGDB_C012056PGDB_AS002062View
2D structure for PGDB_C012141
Dmax-=87.7%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A010135PGDB_C012141PGDB_AS002062View
2D structure for PGDB_C012077
Dmax-=91.3%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A010284PGDB_C012077PGDB_AS002062View
2D structure for PGDB_C012159
Dmax-=89.1%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A010328PGDB_C012159PGDB_AS002062View
2D structure for PGDB_C012110
Dmax-=92%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A010751PGDB_C012110PGDB_AS002062View
2D structure for PGDB_C012116
Dmax-=92.9%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A011068PGDB_C012116PGDB_AS002062View
2D structure for PGDB_C012073
Dmax-=79.5%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A011238PGDB_C012073PGDB_AS002062View
2D structure for PGDB_C012099
Dmax-=93.3%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A011443PGDB_C012099PGDB_AS002062View
2D structure for PGDB_C012146
Dmax-=89.6%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A012171PGDB_C012146PGDB_AS002062View
2D structure for PGDB_C012083
Dmax-=87.5%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A012293PGDB_C012083PGDB_AS002062View
2D structure for PGDB_C012121
Dmax-=90.5%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A012741PGDB_C012121PGDB_AS002062View
2D structure for PGDB_C012094
Dmax-=92.3%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A012841PGDB_C012094PGDB_AS002062View
2D structure for PGDB_C012088
Dmax-=95%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A013339PGDB_C012088PGDB_AS002062View
2D structure for PGDB_C012060
Dmax-=79.9%Concentration series: 10 uM, 0.316 nM20 hWIZ-HT-1080WO2025256460A1PGDB_A013770PGDB_C012060PGDB_AS002062View