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Compound
PGDB_C012127
2 activity records1 related patents
2D structure
CCn1cc(F)c(N2CCC(CN3CCN(Cc4ccn5nc(F)c(N6CCC(=O)NC6=O)c5c4)C[C@@H]3C)CC2)n1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 93.5 | % | Concentration series: 10 uM, 0.316 nM | 20 h | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A008834 | PGDB_C012127 | PGDB_AS002062 | View |
| DC50 | - | = | 22.5 | nM | - | — | WIZ | - | HT-1080 | WO2025256460A1 | PGDB_A045311 | PGDB_C012127 | PGDB_AS000508 | View |