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Compound
PGDB_C015358
5 activity records2 related patents
2D structure
O=C1CCC(N2C(=O)c3cccc4c(Cc5cnn(C6CCN(C(=O)C7(C(F)(F)F)CCC7)CC6)c5)ccc2c34)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | < | 45 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | > 100 nM | - | - | KELLY.2 | WO2022081927A1 | PGDB_A024507 | PGDB_C015358 | PGDB_AS000499 | View |
| DC50 | - | > | 10000 | nM | - | — | - | - | 293T.114 | WO2022081927A1 | PGDB_A033538 | PGDB_C015358 | PGDB_AS001223 | View |
| Emax | - | > | 95 | % | - | DC50 > 10000 nM | > 100 nM | DC50 < 100 nM | - | - | 293T.114 | WO2022081927A1 | PGDB_A037949 | PGDB_C015358 | PGDB_AS000287 | View |
| DC50 | - | < | 100 | nM | - | — | - | - | KELLY.2 | WO2022081927A1 | PGDB_A063022 | PGDB_C015358 | PGDB_AS001296 | View |
| IC50 | - | < | 1 | nM | - | — | - | - | NCI-H929 | EA048567B1 | PGDB_A064201 | PGDB_C015358 | PGDB_AS000893 | View |