Assay

PGDB_AS000287

System: cell_basedTarget: GSPT1Cell line: 293T.114
Assay context summary

Assay context

30 activity records
Assay family% Degradation
Systemcell_based
ReadoutEmax
TargetGSPT1
E3Not specified
Cell line293T.114
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

30 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C016636
Emax->=45%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A007521PGDB_C016636PGDB_AS000287View
2D structure for PGDB_C016638
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A009296PGDB_C016638PGDB_AS000287View
2D structure for PGDB_C016642
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A009578PGDB_C016642PGDB_AS000287View
2D structure for PGDB_C026783
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A012033PGDB_C026783PGDB_AS000287View
2D structure for PGDB_C016651
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A015247PGDB_C016651PGDB_AS000287View
2D structure for PGDB_C026778
Emax->=45%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A015911PGDB_C026778PGDB_AS000287View
2D structure for PGDB_C019149
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A016011PGDB_C019149PGDB_AS000287View
2D structure for PGDB_C016641
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A017332PGDB_C016641PGDB_AS000287View
2D structure for PGDB_C026764
Emax-<45%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A017352PGDB_C026764PGDB_AS000287View
2D structure for PGDB_C016639
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A018496PGDB_C016639PGDB_AS000287View
2D structure for PGDB_C025110
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A022464PGDB_C025110PGDB_AS000287View
2D structure for PGDB_C016640
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A023965PGDB_C016640PGDB_AS000287View
2D structure for PGDB_C016649
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A026691PGDB_C016649PGDB_AS000287View
2D structure for PGDB_C016650
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A026859PGDB_C016650PGDB_AS000287View
2D structure for PGDB_C015421
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A027885PGDB_C015421PGDB_AS000287View
2D structure for PGDB_C016652
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A033757PGDB_C016652PGDB_AS000287View
2D structure for PGDB_C015358
Emax->95%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A037949PGDB_C015358PGDB_AS000287View
2D structure for PGDB_C026785
Emax->95%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A038776PGDB_C026785PGDB_AS000287View
2D structure for PGDB_C016634
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A044469PGDB_C016634PGDB_AS000287View
2D structure for PGDB_C015373
Emax->60%-DC50 > 10000 nM | > 100 nM | DC50 < 100 nM--293T.114WO2022081927A1PGDB_A047412PGDB_C015373PGDB_AS000287View
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