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SIMM · NJU
Assay
PGDB_AS001223
System: cell_based
Target: GSPT1
Cell line: 293T.114
Assay context summary
Assay context
30 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
GSPT1
E3
Not specified
Cell line
293T.114
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
30 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A011907
PGDB_C016638
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A014576
PGDB_C016639
PGDB_AS001223
View
DC50
-
>
100
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A016760
PGDB_C016643
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A017117
PGDB_C016649
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A019867
PGDB_C016653
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A020297
PGDB_C026783
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A021665
PGDB_C016636
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A023131
PGDB_C025110
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A023622
PGDB_C016630
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A024232
PGDB_C016632
PGDB_AS001223
View
DC50
-
>
100
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A024869
PGDB_C016640
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A033538
PGDB_C015358
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A036017
PGDB_C015421
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A037705
PGDB_C026791
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A038745
PGDB_C026778
PGDB_AS001223
View
DC50
-
>
100
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A041326
PGDB_C016651
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A042988
PGDB_C026790
PGDB_AS001223
View
DC50
-
<
100
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A043787
PGDB_C026764
PGDB_AS001223
View
DC50
-
>
10000
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A044954
PGDB_C024947
PGDB_AS001223
View
DC50
-
>
100
nM
-
—
-
-
293T.114
WO2022081927A1
PGDB_A050284
PGDB_C019149
PGDB_AS001223
View