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Compound
PGDB_C016649
4 activity records1 related patents
2D structure
Cc1ccc(CN2CCC(c3ccc4c5c(cccc35)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1FCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | > | 10000 | nM | - | — | - | - | 293T.114 | WO2022081927A1 | PGDB_A017117 | PGDB_C016649 | PGDB_AS001223 | View |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | > 100 nM | DC50 < 100 nM | - | - | 293T.114 | WO2022081927A1 | PGDB_A026691 | PGDB_C016649 | PGDB_AS000287 | View |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | > 100 nM | - | - | KELLY.2 | WO2022081927A1 | PGDB_A036922 | PGDB_C016649 | PGDB_AS000499 | View |
| DC50 | - | > | 10000 | nM | - | — | - | - | KELLY.2 | WO2022081927A1 | PGDB_A042627 | PGDB_C016649 | PGDB_AS001296 | View |