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Compound
PGDB_C019171
4 activity records1 related patents
2D structure
COc1ncc(CN2CCC(c3ccc4c5c(ccnc35)N(C3CCC(=O)NC3=O)C4=O)CC2)cn1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | > | 10000 | nM | - | — | IKZF2 | - | JURKAT.21 | AU2021361043A9 | PGDB_A012677 | PGDB_C019171 | PGDB_AS000724 | View |
| Emax | - | = | 60-95 | % | 10 uM | DC50 > 10000 nM | IKZF2 | - | JURKAT.21 | AU2021361043A9 | PGDB_A046413 | PGDB_C019171 | PGDB_AS001733 | View |
| DC50 | - | > | 10000 | nM | - | — | GSPT1 | - | 293T.114 | AU2021361043A9 | PGDB_A052846 | PGDB_C019171 | PGDB_AS002445 | View |
| Emax | - | > | 95 | % | 10 uM | DC50 > 10000 nM | GSPT1 | - | 293T.114 | AU2021361043A9 | PGDB_A055060 | PGDB_C019171 | PGDB_AS000916 | View |