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SIMM · NJU
Assay
PGDB_AS000916
System: cell_based
Target: GSPT1
Cell line: 293T.114
Assay context summary
Assay context
21 activity records
Assay family
% Degradation
System
cell_based
Readout
Emax
Target
GSPT1
E3
Not specified
Cell line
293T.114
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
21 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A008798
PGDB_C016642
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A010699
PGDB_C019162
PGDB_AS000916
View
Emax
-
>
95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A011049
PGDB_C019154
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A022671
PGDB_C019168
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A024211
PGDB_C019169
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A026298
PGDB_C016641
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A029024
PGDB_C019164
PGDB_AS000916
View
Emax
-
>
95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A030955
PGDB_C019157
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A036661
PGDB_C019153
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A037771
PGDB_C019152
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A039884
PGDB_C019159
PGDB_AS000916
View
Emax
-
>
95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A040818
PGDB_C019155
PGDB_AS000916
View
Emax
-
>
95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A055060
PGDB_C019171
PGDB_AS000916
View
Emax
-
>
95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A057489
PGDB_C019156
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A059118
PGDB_C019165
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A062195
PGDB_C016643
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A063280
PGDB_C019149
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A065271
PGDB_C019161
PGDB_AS000916
View
Emax
-
>
95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A072577
PGDB_C019160
PGDB_AS000916
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
GSPT1
-
293T.114
AU2021361043A9
PGDB_A073996
PGDB_C016651
PGDB_AS000916
View