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SIMM · NJU
Assay
PGDB_AS001733
System: cell_based
Target: IKZF2
Cell line: JURKAT.21
Assay context summary
Assay context
21 activity records
Assay family
% Degradation
System
cell_based
Readout
Emax
Target
IKZF2
E3
Not specified
Cell line
JURKAT.21
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
21 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A009073
PGDB_C019158
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A009903
PGDB_C019167
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A012609
PGDB_C016643
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A012775
PGDB_C016651
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A015038
PGDB_C019157
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A015467
PGDB_C019164
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A017454
PGDB_C019152
PGDB_AS001733
View
Emax
-
>
95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A020206
PGDB_C019169
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A022515
PGDB_C019155
PGDB_AS001733
View
Emax
-
=
45-60
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A026172
PGDB_C016642
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A027542
PGDB_C019154
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A031650
PGDB_C019161
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A040720
PGDB_C019153
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A046413
PGDB_C019171
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A050643
PGDB_C019168
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A051845
PGDB_C019156
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A055181
PGDB_C019159
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A059867
PGDB_C019166
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A074365
PGDB_C019163
PGDB_AS001733
View
Emax
-
=
60-95
%
10 uM
DC50 > 10000 nM
IKZF2
-
JURKAT.21
AU2021361043A9
PGDB_A075745
PGDB_C019160
PGDB_AS001733
View