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O=C1CCC(N2Cc3cc(CN4CCC(c5noc6cc(F)ccc56)CC4)c(F)cc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 10-50 | nM | - | — | IKZF3 | - | TMD8 | WO2025016359A1 | PGDB_A032713 | PGDB_C019539 | PGDB_AS000926 | View | |
| IC50 | - | = | 1-5 | nM | - | — | IKZF3 | - | MOLT-4 | WO2025016359A1 | PGDB_A046357 | PGDB_C019539 | PGDB_AS001975 | View | |
| IC50 | - | = | 10-50 | nM | - | — | IKZF3 | - | H1975 | WO2025016359A1 | PGDB_A050635 | PGDB_C019539 | PGDB_AS000939 | View | |
| IC50 | - | = | 10-50 | nM | - | — | IKZF3 | - | MDA-MB-231 | WO2025016359A1 | PGDB_A056069 | PGDB_C019539 | PGDB_AS000537 | View | |
| IC50 | - | = | 1.5-1.9 | uM | - | — | CRBN | CRBN | - | WO2025016359A1 | PGDB_A062147 | PGDB_C019539 | PGDB_AS001897 | View |