Assay

PGDB_AS001897

System: biochemicalTarget: CRBN
Assay context summary

Assay context

254 activity records
Assay familybiochemical
Systembiochemical
ReadoutIC50
TargetCRBN
E3CRBN
OrganismHomo sapiens
TechnologyHTRF
Activity compounds and values

Activity records

254 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019294
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A007436PGDB_C019294PGDB_AS001897View
2D structure for PGDB_C019482
IC50-=0.5-1uM-—CRBNCRBN-WO2025016359A1PGDB_A007871PGDB_C019482PGDB_AS001897View
2D structure for PGDB_C019387
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A008636PGDB_C019387PGDB_AS001897View
2D structure for PGDB_C019322
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A008705PGDB_C019322PGDB_AS001897View
2D structure for PGDB_C019331
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A009040PGDB_C019331PGDB_AS001897View
2D structure for PGDB_C019537
IC50-=1-1.5uM-—CRBNCRBN-WO2025016359A1PGDB_A009255PGDB_C019537PGDB_AS001897View
2D structure for PGDB_C019202
IC50-=0.5-1uM-—CRBNCRBN-WO2025016359A1PGDB_A009987PGDB_C019202PGDB_AS001897View
2D structure for PGDB_C019359
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A009992PGDB_C019359PGDB_AS001897View
2D structure for PGDB_C019309
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A010117PGDB_C019309PGDB_AS001897View
2D structure for PGDB_C019310
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A010223PGDB_C019310PGDB_AS001897View
2D structure for PGDB_C019220
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A010416PGDB_C019220PGDB_AS001897View
2D structure for PGDB_C019538
IC50-=1-1.5uM-—CRBNCRBN-WO2025016359A1PGDB_A011162PGDB_C019538PGDB_AS001897View
2D structure for PGDB_C019225
IC50-=0.5-1uM-—CRBNCRBN-WO2025016359A1PGDB_A011237PGDB_C019225PGDB_AS001897View
2D structure for PGDB_C019285
IC50-=1-1.5uM-—CRBNCRBN-WO2025016359A1PGDB_A011299PGDB_C019285PGDB_AS001897View
2D structure for PGDB_C019411
IC50-=1.5-1.9uM-—CRBNCRBN-WO2025016359A1PGDB_A011624PGDB_C019411PGDB_AS001897View
2D structure for PGDB_C019377
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A011712PGDB_C019377PGDB_AS001897View
2D structure for PGDB_C019197
IC50-=0.5-1uM-—CRBNCRBN-WO2025016359A1PGDB_A011886PGDB_C019197PGDB_AS001897View
2D structure for PGDB_C019246
IC50-=0.5-1uM-—CRBNCRBN-WO2025016359A1PGDB_A011946PGDB_C019246PGDB_AS001897View
2D structure for PGDB_C019384
IC50-<=0.5uM-—CRBNCRBN-WO2025016359A1PGDB_A012257PGDB_C019384PGDB_AS001897View
2D structure for PGDB_C019362
IC50-=0.5-1uM-—CRBNCRBN-WO2025016359A1PGDB_A012676PGDB_C019362PGDB_AS001897View
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