Assay context summary

Assay context

33 activity records
Activity compounds and values

Activity records

33 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019331
IC50-=50-100nM-IKZF3-TMD8WO2025016359A1PGDB_A007109PGDB_C019331PGDB_AS000926View
2D structure for PGDB_C019261
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A014372PGDB_C019261PGDB_AS000926View
2D structure for PGDB_C019270
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A015472PGDB_C019270PGDB_AS000926View
2D structure for PGDB_C019272
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A016203PGDB_C019272PGDB_AS000926View
2D structure for PGDB_C019286
IC50-=500-1000nM-IKZF3-TMD8WO2025016359A1PGDB_A016935PGDB_C019286PGDB_AS000926View
2D structure for PGDB_C019275
IC50-=500-1000nM-IKZF3-TMD8WO2025016359A1PGDB_A017351PGDB_C019275PGDB_AS000926View
2D structure for PGDB_C019175
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A018080PGDB_C019175PGDB_AS000926View
2D structure for PGDB_C019334
IC50-=500-1000nM-IKZF3-TMD8WO2025016359A1PGDB_A021262PGDB_C019334PGDB_AS000926View
2D structure for PGDB_C019315
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A027077PGDB_C019315PGDB_AS000926View
2D structure for PGDB_C019316
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A029551PGDB_C019316PGDB_AS000926View
2D structure for PGDB_C019264
IC50-=50-100nM-IKZF3-TMD8WO2025016359A1PGDB_A030316PGDB_C019264PGDB_AS000926View
2D structure for PGDB_C019287
IC50-=100-500nM-IKZF3-TMD8WO2025016359A1PGDB_A031782PGDB_C019287PGDB_AS000926View
2D structure for PGDB_C019323
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A032318PGDB_C019323PGDB_AS000926View
2D structure for PGDB_C019539
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A032713PGDB_C019539PGDB_AS000926View
2D structure for PGDB_C019274
IC50-=500-1000nM-IKZF3-TMD8WO2025016359A1PGDB_A034907PGDB_C019274PGDB_AS000926View
2D structure for PGDB_C019330
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A036254PGDB_C019330PGDB_AS000926View
2D structure for PGDB_C019296
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A036921PGDB_C019296PGDB_AS000926View
2D structure for PGDB_C019177
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A037116PGDB_C019177PGDB_AS000926View
2D structure for PGDB_C019263
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A040705PGDB_C019263PGDB_AS000926View
2D structure for PGDB_C019290
IC50-=10-50nM-IKZF3-TMD8WO2025016359A1PGDB_A042450PGDB_C019290PGDB_AS000926View