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Compound
PGDB_C020485
3 activity records1 related patents
2D structure
CNCC1(COCCc2ccc(C(Cl)NCc3ccc4c5c(cccc35)C(=O)N4C3CCC(=O)NC3=O)cc2Cl)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.5-5 | nM | - | — | GSPT1 | - | HEK293T | WO2025162410A1 | PGDB_A012120 | PGDB_C020485 | PGDB_AS002143 | View |
| EC50 | - | = | 0.5-5 | nM | - | — | GSPT1 | - | - | WO2025162410A1 | PGDB_A068207 | PGDB_C020485 | PGDB_AS002258 | View |
| Selectivity index | 293T/HCC569 | >= | 100 | fold | - | — | - | - | - | WO2025162410A1 | PGDB_A072992 | PGDB_C020485 | PGDB_AS000299 | View |