Assay

PGDB_AS002258

System: cell_basedTarget: GSPT1
Assay context summary

Assay context

68 activity records
Assay family% Degradation
Systemcell_based
ReadoutEC50
TargetGSPT1
E3Not specified
OrganismHomo sapiens
Technologyfluorescence
Activity compounds and values

Activity records

68 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020477
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A008456PGDB_C020477PGDB_AS002258View
2D structure for PGDB_C020478
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A009253PGDB_C020478PGDB_AS002258View
2D structure for PGDB_C020490
EC50->5nM-—GSPT1--WO2025162410A1PGDB_A011593PGDB_C020490PGDB_AS002258View
2D structure for PGDB_C020500
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A013000PGDB_C020500PGDB_AS002258View
2D structure for PGDB_C020477
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A013334PGDB_C020477PGDB_AS002258View
2D structure for PGDB_C020475
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A013349PGDB_C020475PGDB_AS002258View
2D structure for PGDB_C020496
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A014193PGDB_C020496PGDB_AS002258View
2D structure for PGDB_C020471
EC50-=0.5-5nM-—GSPT1--WO2025162410A1PGDB_A016958PGDB_C020471PGDB_AS002258View
2D structure for PGDB_C020497
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A018465PGDB_C020497PGDB_AS002258View
2D structure for PGDB_C020474
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A020088PGDB_C020474PGDB_AS002258View
2D structure for PGDB_C020482
EC50->5nM-—GSPT1--WO2025162410A1PGDB_A020868PGDB_C020482PGDB_AS002258View
2D structure for PGDB_C020487
EC50->5nM-—GSPT1--WO2025162410A1PGDB_A020911PGDB_C020487PGDB_AS002258View
2D structure for PGDB_C020461
EC50-=0.5-5nM-—GSPT1--WO2025162410A1PGDB_A021965PGDB_C020461PGDB_AS002258View
2D structure for PGDB_C020476
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A022547PGDB_C020476PGDB_AS002258View
2D structure for PGDB_C020495
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A023373PGDB_C020495PGDB_AS002258View
2D structure for PGDB_C020504
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A025207PGDB_C020504PGDB_AS002258View
2D structure for PGDB_C020464
EC50->5nM-—GSPT1--WO2025162410A1PGDB_A025321PGDB_C020464PGDB_AS002258View
2D structure for PGDB_C020467
EC50-=0.5-5nM-—GSPT1--WO2025162410A1PGDB_A026313PGDB_C020467PGDB_AS002258View
2D structure for PGDB_C020498
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A027914PGDB_C020498PGDB_AS002258View
2D structure for PGDB_C020481
EC50-=<= 0.5nM-—GSPT1--WO2025162410A1PGDB_A028713PGDB_C020481PGDB_AS002258View
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