Assay context summary

Assay context

68 activity records
Activity compounds and values

Activity records

68 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020503
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A007269PGDB_C020503PGDB_AS002143View
2D structure for PGDB_C020481
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A007505PGDB_C020481PGDB_AS002143View
2D structure for PGDB_C020499
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A007633PGDB_C020499PGDB_AS002143View
2D structure for PGDB_C020469
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A009655PGDB_C020469PGDB_AS002143View
2D structure for PGDB_C020462
IC50->5nM-GSPT1-HEK293TWO2025162410A1PGDB_A011798PGDB_C020462PGDB_AS002143View
2D structure for PGDB_C020485
IC50-=0.5-5nM-GSPT1-HEK293TWO2025162410A1PGDB_A012120PGDB_C020485PGDB_AS002143View
2D structure for PGDB_C020504
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A012648PGDB_C020504PGDB_AS002143View
2D structure for PGDB_C020486
IC50->5nM-GSPT1-HEK293TWO2025162410A1PGDB_A013264PGDB_C020486PGDB_AS002143View
2D structure for PGDB_C020484
IC50-=0.5-5nM-GSPT1-HEK293TWO2025162410A1PGDB_A013422PGDB_C020484PGDB_AS002143View
2D structure for PGDB_C020504
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A014428PGDB_C020504PGDB_AS002143View
2D structure for PGDB_C020495
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A017076PGDB_C020495PGDB_AS002143View
2D structure for PGDB_C020475
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A017241PGDB_C020475PGDB_AS002143View
2D structure for PGDB_C020489
IC50->5nM-GSPT1-HEK293TWO2025162410A1PGDB_A017371PGDB_C020489PGDB_AS002143View
2D structure for PGDB_C020472
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A017503PGDB_C020472PGDB_AS002143View
2D structure for PGDB_C020480
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A017893PGDB_C020480PGDB_AS002143View
2D structure for PGDB_C020492
IC50-=0.5-5nM-GSPT1-HEK293TWO2025162410A1PGDB_A018761PGDB_C020492PGDB_AS002143View
2D structure for PGDB_C020502
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A020480PGDB_C020502PGDB_AS002143View
2D structure for PGDB_C020476
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A020903PGDB_C020476PGDB_AS002143View
2D structure for PGDB_C020475
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A021939PGDB_C020475PGDB_AS002143View
2D structure for PGDB_C020497
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A022597PGDB_C020497PGDB_AS002143View