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Compound
PGDB_C023741
10 activity records1 related patents
2D structure
Cc1sc2ncnc(C3=CCN(Cc4ccc5c(c4)CN(N4CCC(=O)NC4=O)C5=O)CC3)c2c1CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 15-20 | % | 10 nM | - | - | - | H292 | WO2024245444A1 | PGDB_A023539 | PGDB_C023741 | PGDB_AS001605 | View |
| % Inhibition | - | = | 20-40 | % | 500 nM | - | - | - | H292 | WO2024245444A1 | PGDB_A024368 | PGDB_C023741 | PGDB_AS000415 | View |
| % Inhibition | - | = | 60-80 | % | 500 nM | - | - | - | MM.1S | WO2024245444A1 | PGDB_A025462 | PGDB_C023741 | PGDB_AS000503 | View |
| % Inhibition | - | = | 80-100 | % | 500 nM | - | - | - | MV-4-11 | WO2024245444A1 | PGDB_A031424 | PGDB_C023741 | PGDB_AS000199 | View |
| % Inhibition | - | = | 25-30 | % | 500 nM | - | - | - | H2228 | WO2024245444A1 | PGDB_A033783 | PGDB_C023741 | PGDB_AS000051 | View |
| % Inhibition | - | < | 5 | % | 10 nM | - | - | - | MM.1S | WO2024245444A1 | PGDB_A043926 | PGDB_C023741 | PGDB_AS001568 | View |
| % Inhibition | - | = | 30-40 | % | 10 nM | - | - | - | MV-4-11 | WO2024245444A1 | PGDB_A055401 | PGDB_C023741 | PGDB_AS001519 | View |
| % Inhibition | - | = | 10-15 | % | 10 nM | - | - | - | MDA-MB-231 | WO2024245444A1 | PGDB_A066553 | PGDB_C023741 | PGDB_AS002156 | View |
| % Inhibition | - | = | 18-25 | % | 500 nM | - | - | - | MDA-MB-231 | WO2024245444A1 | PGDB_A070168 | PGDB_C023741 | PGDB_AS002131 | View |
| % Inhibition | - | = | 10-15 | % | 10 nM | - | - | - | H2228 | WO2024245444A1 | PGDB_A073854 | PGDB_C023741 | PGDB_AS001356 | View |