Assay context summary

Assay context

36 activity records
Activity compounds and values

Activity records

36 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C023621
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A008422PGDB_C023621PGDB_AS000051View
2D structure for PGDB_C014263
% Inhibition-=30-40%500 nM---H2228WO2024245444A1PGDB_A012404PGDB_C014263PGDB_AS000051View
2D structure for PGDB_C014203
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A019745PGDB_C014203PGDB_AS000051View
2D structure for PGDB_C014279
% Inhibition-=25-30%500 nM---H2228WO2024245444A1PGDB_A020370PGDB_C014279PGDB_AS000051View
2D structure for PGDB_C014278
% Inhibition-=25-30%500 nM---H2228WO2024245444A1PGDB_A020382PGDB_C014278PGDB_AS000051View
2D structure for PGDB_C014262
% Inhibition-=15-20%500 nM---H2228WO2024245444A1PGDB_A025627PGDB_C014262PGDB_AS000051View
2D structure for PGDB_C014308
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A026610PGDB_C014308PGDB_AS000051View
2D structure for PGDB_C014326
% Inhibition-=25-30%500 nM---H2228WO2024245444A1PGDB_A029005PGDB_C014326PGDB_AS000051View
2D structure for PGDB_C014259
% Inhibition-=30-40%500 nM---H2228WO2024245444A1PGDB_A029087PGDB_C014259PGDB_AS000051View
2D structure for PGDB_C014202
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A029274PGDB_C014202PGDB_AS000051View
2D structure for PGDB_C023741
% Inhibition-=25-30%500 nM---H2228WO2024245444A1PGDB_A033783PGDB_C023741PGDB_AS000051View
2D structure for PGDB_C014271
% Inhibition-=30-40%500 nM---H2228WO2024245444A1PGDB_A034281PGDB_C014271PGDB_AS000051View
2D structure for PGDB_C014260
% Inhibition-=25-30%500 nM---H2228WO2024245444A1PGDB_A034483PGDB_C014260PGDB_AS000051View
2D structure for PGDB_C014270
% Inhibition-=25-30%500 nM---H2228WO2024245444A1PGDB_A035034PGDB_C014270PGDB_AS000051View
2D structure for PGDB_C014306
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A038543PGDB_C014306PGDB_AS000051View
2D structure for PGDB_C014307
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A038763PGDB_C014307PGDB_AS000051View
2D structure for PGDB_C023633
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A040607PGDB_C023633PGDB_AS000051View
2D structure for PGDB_C014200
% Inhibition-=25-30%500 nM---H2228WO2024245444A1PGDB_A043009PGDB_C014200PGDB_AS000051View
2D structure for PGDB_C014309
% Inhibition-=20-25%500 nM---H2228WO2024245444A1PGDB_A044023PGDB_C014309PGDB_AS000051View
2D structure for PGDB_C014264
% Inhibition-=30-40%500 nM---H2228WO2024245444A1PGDB_A044501PGDB_C014264PGDB_AS000051View