Assay context summary

Assay context

36 activity records
Activity compounds and values

Activity records

36 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C014278
% Inhibition-=15-20%10 nM---H2228WO2024245444A1PGDB_A008087PGDB_C014278PGDB_AS001356View
2D structure for PGDB_C014306
% Inhibition-=20-25%10 nM---H2228WO2024245444A1PGDB_A010709PGDB_C014306PGDB_AS001356View
2D structure for PGDB_C023714
% Inhibition-=25-30%10 nM---H2228WO2024245444A1PGDB_A014382PGDB_C023714PGDB_AS001356View
2D structure for PGDB_C023633
% Inhibition-=15-20%10 nM---H2228WO2024245444A1PGDB_A020175PGDB_C023633PGDB_AS001356View
2D structure for PGDB_C014312
% Inhibition-=15-20%10 nM---H2228WO2024245444A1PGDB_A021895PGDB_C014312PGDB_AS001356View
2D structure for PGDB_C014260
% Inhibition-=10-15%10 nM---H2228WO2024245444A1PGDB_A023653PGDB_C014260PGDB_AS001356View
2D structure for PGDB_C023632
% Inhibition-=5-10%10 nM---H2228WO2024245444A1PGDB_A024543PGDB_C023632PGDB_AS001356View
2D structure for PGDB_C014263
% Inhibition-=20-25%10 nM---H2228WO2024245444A1PGDB_A024688PGDB_C014263PGDB_AS001356View
2D structure for PGDB_C014203
% Inhibition-=30-40%10 nM---H2228WO2024245444A1PGDB_A028343PGDB_C014203PGDB_AS001356View
2D structure for PGDB_C014309
% Inhibition-=20-25%10 nM---H2228WO2024245444A1PGDB_A029499PGDB_C014309PGDB_AS001356View
2D structure for PGDB_C023620
% Inhibition-=20-25%10 nM---H2228WO2024245444A1PGDB_A036899PGDB_C023620PGDB_AS001356View
2D structure for PGDB_C014262
% Inhibition-=30-40%10 nM---H2228WO2024245444A1PGDB_A037182PGDB_C014262PGDB_AS001356View
2D structure for PGDB_C014264
% Inhibition-=25-30%10 nM---H2228WO2024245444A1PGDB_A038338PGDB_C014264PGDB_AS001356View
2D structure for PGDB_C014273
% Inhibition-=25-30%10 nM---H2228WO2024245444A1PGDB_A038917PGDB_C014273PGDB_AS001356View
2D structure for PGDB_C014259
% Inhibition-=25-30%10 nM---H2228WO2024245444A1PGDB_A039167PGDB_C014259PGDB_AS001356View
2D structure for PGDB_C014307
% Inhibition-=20-25%10 nM---H2228WO2024245444A1PGDB_A040823PGDB_C014307PGDB_AS001356View
2D structure for PGDB_C014261
% Inhibition-=30-40%10 nM---H2228WO2024245444A1PGDB_A043006PGDB_C014261PGDB_AS001356View
2D structure for PGDB_C014308
% Inhibition-=20-25%10 nM---H2228WO2024245444A1PGDB_A043519PGDB_C014308PGDB_AS001356View
2D structure for PGDB_C014327
% Inhibition-=10-15%10 nM---H2228WO2024245444A1PGDB_A044829PGDB_C014327PGDB_AS001356View
2D structure for PGDB_C014268
% Inhibition-=25-30%10 nM---H2228WO2024245444A1PGDB_A045124PGDB_C014268PGDB_AS001356View