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Compound
PGDB_C024458
6 activity records1 related patents
2D structure
COc1cc(CN2CCN(Nc3ccc4c(c3F)CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 20-30 | % | 0.1 uM | - | IKZF3 | - | - | WO2025162225A1 | PGDB_A011318 | PGDB_C024458 | PGDB_AS000994 | View |
| % Inhibition | - | = | 70-80 | % | 2 uM | - | CRBN | CRBN | - | WO2025162225A1 | PGDB_A035104 | PGDB_C024458 | PGDB_AS002540 | View |
| % Inhibition | - | = | 20-30 | % | 0.1 uM | - | IKZF3 | - | - | WO2025162225A1 | PGDB_A039362 | PGDB_C024458 | PGDB_AS002324 | View |
| % Inhibition | - | = | 0-10 | % | 0.1 uM | - | IKZF3 | - | - | WO2025162225A1 | PGDB_A049344 | PGDB_C024458 | PGDB_AS002550 | View |
| % Inhibition | - | = | 0-10 | % | 0.1 uM | - | IKZF3 | - | - | WO2025162225A1 | PGDB_A064154 | PGDB_C024458 | PGDB_AS000702 | View |
| % Inhibition | - | = | 40-53 | % | 0.5 uM | - | CRBN | CRBN | - | WO2025162225A1 | PGDB_A065740 | PGDB_C024458 | PGDB_AS002133 | View |