Assay

PGDB_AS002540

System: cell_basedTarget: CRBN
Assay context summary

Assay context

239 activity records
Assay familybiochemical
Systemcell_based
Readout% Inhibition
TargetCRBN
E3CRBN
TechnologyHTRF
Detection targetcell_inhibition
Activity compounds and values

Activity records

239 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C024512
% Inhibition-=53-60%2 uM-CRBNCRBN-WO2025162225A1PGDB_A007006PGDB_C024512PGDB_AS002540View
2D structure for PGDB_C024353
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A007404PGDB_C024353PGDB_AS002540View
2D structure for PGDB_C024211
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A007461PGDB_C024211PGDB_AS002540View
2D structure for PGDB_C024504
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A007696PGDB_C024504PGDB_AS002540View
2D structure for PGDB_C024527
% Inhibition-=60-70%2 uM-CRBNCRBN-WO2025162225A1PGDB_A008014PGDB_C024527PGDB_AS002540View
2D structure for PGDB_C024482
% Inhibition-=70-80%2 uM-CRBNCRBN-WO2025162225A1PGDB_A008586PGDB_C024482PGDB_AS002540View
2D structure for PGDB_C024433
% Inhibition-=60-70%2 uM-CRBNCRBN-WO2025162225A1PGDB_A009484PGDB_C024433PGDB_AS002540View
2D structure for PGDB_C024493
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A010061PGDB_C024493PGDB_AS002540View
2D structure for PGDB_C024358
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A010546PGDB_C024358PGDB_AS002540View
2D structure for PGDB_C024223
% Inhibition-=60-70%2 uM-CRBNCRBN-WO2025162225A1PGDB_A010928PGDB_C024223PGDB_AS002540View
2D structure for PGDB_C024476
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A010964PGDB_C024476PGDB_AS002540View
2D structure for PGDB_C024521
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A010965PGDB_C024521PGDB_AS002540View
2D structure for PGDB_C024369
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A011399PGDB_C024369PGDB_AS002540View
2D structure for PGDB_C024510
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A012344PGDB_C024510PGDB_AS002540View
2D structure for PGDB_C024235
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A012475PGDB_C024235PGDB_AS002540View
2D structure for PGDB_C024230
% Inhibition-=60-70%2 uM-CRBNCRBN-WO2025162225A1PGDB_A012491PGDB_C024230PGDB_AS002540View
2D structure for PGDB_C024532
% Inhibition-=70-80%2 uM-CRBNCRBN-WO2025162225A1PGDB_A012601PGDB_C024532PGDB_AS002540View
2D structure for PGDB_C024516
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A013011PGDB_C024516PGDB_AS002540View
2D structure for PGDB_C024246
% Inhibition-=70-80%2 uM-CRBNCRBN-WO2025162225A1PGDB_A013191PGDB_C024246PGDB_AS002540View
2D structure for PGDB_C024350
% Inhibition-=80-100%2 uM-CRBNCRBN-WO2025162225A1PGDB_A013239PGDB_C024350PGDB_AS002540View
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