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O=C1CCC(N2Cc3cc(CN4CCC(n5cc(NC(=O)c6cnn7ccc(N8CCOCC8)nc67)c(C(F)F)n5)CC4)cc(F)c3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | Mino | CN116239566A | PGDB_A017163 | PGDB_C025956 | PGDB_AS000456 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A043856 | PGDB_C025956 | PGDB_AS000709 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | IRAK4 | - | SU-DHL-4 | CN116239566A | PGDB_A064967 | PGDB_C025956 | PGDB_AS002569 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | IRAK4 | - | SW620 | CN116239566A | PGDB_A069537 | PGDB_C025956 | PGDB_AS000233 | View |