Assay
PGDB_AS000456
System: cell_basedCell line: Mino
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Mino | CN116239566A | PGDB_A014113 | PGDB_C019639 | PGDB_AS000456 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | Mino | CN116239566A | PGDB_A017163 | PGDB_C025956 | PGDB_AS000456 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | IRAK4 | - | Mino | CN116239566A | PGDB_A021464 | PGDB_C019640 | PGDB_AS000456 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Mino | CN116239566A | PGDB_A042253 | PGDB_C025954 | PGDB_AS000456 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Mino | CN116239566A | PGDB_A077769 | PGDB_C025953 | PGDB_AS000456 | View |