Assay
PGDB_AS000709
System: cell_basedCell line: MV-4-11
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A007813 | PGDB_C025977 | PGDB_AS000709 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A011355 | PGDB_C025980 | PGDB_AS000709 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A014526 | PGDB_C025954 | PGDB_AS000709 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A018852 | PGDB_C019639 | PGDB_AS000709 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A039749 | PGDB_C025978 | PGDB_AS000709 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A043856 | PGDB_C025956 | PGDB_AS000709 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A047469 | PGDB_C025953 | PGDB_AS000709 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A051375 | PGDB_C019642 | PGDB_AS000709 | View | |
| IC50 | - | = | 50-100 | nM | - | — | IRAK4 | - | MV-4-11 | CN116239566A | PGDB_A066322 | PGDB_C025979 | PGDB_AS000709 | View |