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Compound
PGDB_C027073
4 activity records1 related patents
2D structure
C[C@@H]1CCN(c2cc(-c3ccccc3O)nnc2N)CCN1c1ccnc(C#CCN2CC3(CCC3(F)F)C2)n1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2023244806A1 | PGDB_A009853 | PGDB_C027073 | PGDB_AS000849 | View |
| DC50 | - | = | 0.05-0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2023244806A1 | PGDB_A012938 | PGDB_C027073 | PGDB_AS002237 | View |
| DC50 | - | = | 0.05-0.5 | uM | - | — | SMARCA4 | - | HeLa | WO2023244806A1 | PGDB_A018955 | PGDB_C027073 | PGDB_AS000073 | View |
| % Degradation | - | > | 70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2023244806A1 | PGDB_A052116 | PGDB_C027073 | PGDB_AS001988 | View |