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Compound
PGDB_C027185
4 activity records1 related patents
2D structure
C[C@@H]1CN(CC#Cc2nccc(N3CCCN(c4cc(-c5ccccc5O)nnc4N)CC3)n2)CCO1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 30-70 | % | 1 uM | 24 h | SMARCA2 | - | HeLa | WO2023244806A1 | PGDB_A008678 | PGDB_C027185 | PGDB_AS001988 | View |
| % Degradation | - | < | 30 | % | 1 uM | 24 h | SMARCA4 | - | HeLa | WO2023244806A1 | PGDB_A018836 | PGDB_C027185 | PGDB_AS000849 | View |
| DC50 | - | = | 0.05-0.5 | uM | - | — | SMARCA2 | - | HeLa | WO2023244806A1 | PGDB_A045071 | PGDB_C027185 | PGDB_AS002237 | View |
| DC50 | - | = | 0.5-5 | uM | - | — | SMARCA4 | - | HeLa | WO2023244806A1 | PGDB_A056538 | PGDB_C027185 | PGDB_AS000073 | View |