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Compound
PGDB_C029662
4 activity records1 related patents
2D structure
COC1CCN(C(=O)Nc2c(C)cc(-c3cccc(C4CCC(=O)NC4=O)c3Cl)cc2F)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 0.8 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A000671 | PGDB_C029662 | PGDB_AS001440 | View |
| IC50 | - | < | 0.1 | nM | - | — | VAV1 | - | pan-B | WO2026051943A1 | PGDB_A002050 | PGDB_C029662 | PGDB_AS001700 | View |
| Dmax | - | = | 98.9 | % | Concentration series: 10 uM, 1 uM | - | VAV1 | - | - | WO2026051943A1 | PGDB_A004931 | PGDB_C029662 | PGDB_AS000777 | View |
| IC50 | - | = | 0.0943 | nM | - | — | VAV1 | - | pan-B | WO2026051943A1 | PGDB_A078782 | PGDB_C029662 | PGDB_AS001016 | View |