Assay context summary

Assay context

262 activity records
Activity compounds and values

Activity records

262 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C029586
Dmax-=98.44%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000079PGDB_C029586PGDB_AS000777View
2D structure for PGDB_C029477
Dmax-=98.28%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000133PGDB_C029477PGDB_AS000777View
2D structure for PGDB_C029427
Dmax-=84%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000135PGDB_C029427PGDB_AS000777View
2D structure for PGDB_C029576
Dmax-=98.6%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000152PGDB_C029576PGDB_AS000777View
2D structure for PGDB_C029673
Dmax-=97.3%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000192PGDB_C029673PGDB_AS000777View
2D structure for PGDB_C029444
Dmax-=97.3%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000220PGDB_C029444PGDB_AS000777View
2D structure for PGDB_C029606
Dmax-=98.6%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000224PGDB_C029606PGDB_AS000777View
2D structure for PGDB_C029530
Dmax-=96.58%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000273PGDB_C029530PGDB_AS000777View
2D structure for PGDB_C029491
Dmax-=97.95%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000289PGDB_C029491PGDB_AS000777View
2D structure for PGDB_C029452
Dmax-=97.9%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000294PGDB_C029452PGDB_AS000777View
2D structure for PGDB_C029627
Dmax-=99%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000320PGDB_C029627PGDB_AS000777View
2D structure for PGDB_C029540
Dmax-=98.6%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000479PGDB_C029540PGDB_AS000777View
2D structure for PGDB_C029499
Dmax-=98.07%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000602PGDB_C029499PGDB_AS000777View
2D structure for PGDB_C029617
Dmax-=98.6%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000635PGDB_C029617PGDB_AS000777View
2D structure for PGDB_C029512
Dmax-=98.24%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000640PGDB_C029512PGDB_AS000777View
2D structure for PGDB_C029541
Dmax-=98.62%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000662PGDB_C029541PGDB_AS000777View
2D structure for PGDB_C029622
Dmax-=99%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000667PGDB_C029622PGDB_AS000777View
2D structure for PGDB_C029533
Dmax-=98.37%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000673PGDB_C029533PGDB_AS000777View
2D structure for PGDB_C029650
Dmax-=98.5%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000678PGDB_C029650PGDB_AS000777View
2D structure for PGDB_C029553
Dmax-=98.51%Concentration series: 10 uM, 1 uM-VAV1--WO2026051943A1PGDB_A000701PGDB_C029553PGDB_AS000777View