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Compound
PGDB_C029716
6 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C)(CN5CCC6(CCc7ccc(N8CCC(=O)NC8=O)cc7O6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 94 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000161 | PGDB_C029716 | PGDB_AS001838 | View |
| IC50 | - | = | 0.0025 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A004291 | PGDB_C029716 | PGDB_AS000481 | View |
| % Degradation | - | = | 91 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A006224 | PGDB_C029716 | PGDB_AS002389 | View |
| IC50 | - | = | 0.54 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078933 | PGDB_C029716 | PGDB_AS000195 | View |
| % Degradation | - | = | 76 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080080 | PGDB_C029716 | PGDB_AS002463 | View |
| % Degradation | - | = | 81 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A080462 | PGDB_C029716 | PGDB_AS001354 | View |