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SIMM · NJU
Assay
PGDB_AS002389
System: cell_based
Target: AR
Cell line: LNCaPFGC
Assay context summary
Assay context
431 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
Target
AR
E3
Not specified
Cell line
LNCaPFGC
Organism
Homo sapiens
Technology
Western_blot
Detection target
protein_degradation
Activity compounds and values
Activity records
431 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
=
65
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000006
PGDB_C029932
PGDB_AS002389
View
% Degradation
-
=
93
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000025
PGDB_C029736
PGDB_AS002389
View
% Degradation
-
=
81
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000032
PGDB_C029741
PGDB_AS002389
View
% Degradation
-
=
86
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000035
PGDB_C029794
PGDB_AS002389
View
% Degradation
-
=
40
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000049
PGDB_C029959
PGDB_AS002389
View
% Degradation
-
=
91
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000060
PGDB_C030130
PGDB_AS002389
View
% Degradation
-
=
21
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000073
PGDB_C030116
PGDB_AS002389
View
% Degradation
-
=
79
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000127
PGDB_C029834
PGDB_AS002389
View
% Degradation
-
=
83
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000145
PGDB_C029838
PGDB_AS002389
View
% Degradation
-
=
74
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000174
PGDB_C030003
PGDB_AS002389
View
% Degradation
-
=
84
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000207
PGDB_C030124
PGDB_AS002389
View
% Degradation
-
=
93
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000221
PGDB_C029812
PGDB_AS002389
View
% Degradation
-
=
85
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000300
PGDB_C029920
PGDB_AS002389
View
% Degradation
-
=
72
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000307
PGDB_C029863
PGDB_AS002389
View
% Degradation
-
=
76
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000309
PGDB_C029774
PGDB_AS002389
View
% Degradation
-
=
87
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000316
PGDB_C029859
PGDB_AS002389
View
% Degradation
-
=
92
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000348
PGDB_C030095
PGDB_AS002389
View
% Degradation
-
=
79
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000369
PGDB_C030016
PGDB_AS002389
View
% Degradation
-
=
41
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000416
PGDB_C029719
PGDB_AS002389
View
% Degradation
-
=
77
%
100 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000417
PGDB_C030014
PGDB_AS002389
View