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Compound
PGDB_C029717
6 activity records1 related patents
2D structure
COC1(CN2CCC3(CCc4ccc(N5CCC(=O)NC5=O)cc4O3)CC2)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.017 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A001095 | PGDB_C029717 | PGDB_AS000481 | View |
| IC50 | - | = | 0.64 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A003579 | PGDB_C029717 | PGDB_AS000195 | View |
| % Degradation | - | = | 82 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A006810 | PGDB_C029717 | PGDB_AS002463 | View |
| % Degradation | - | = | 94 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A077994 | PGDB_C029717 | PGDB_AS001838 | View |
| % Degradation | - | = | 88 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A081391 | PGDB_C029717 | PGDB_AS001354 | View |
| % Degradation | - | = | 91 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081729 | PGDB_C029717 | PGDB_AS002389 | View |