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Compound
PGDB_C029722
6 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CCC(N6CCC7(CCc8ccc(N9CCC(=O)NC9=O)cc8O7)CC6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.93 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000456 | PGDB_C029722 | PGDB_AS000195 | View |
| % Degradation | - | = | 50 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001825 | PGDB_C029722 | PGDB_AS002463 | View |
| IC50 | - | = | 0.0065 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A006976 | PGDB_C029722 | PGDB_AS000481 | View |
| % Degradation | - | = | 82 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078932 | PGDB_C029722 | PGDB_AS001838 | View |
| % Degradation | - | = | 81 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079214 | PGDB_C029722 | PGDB_AS002389 | View |
| % Degradation | - | = | 63 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A080158 | PGDB_C029722 | PGDB_AS001354 | View |