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Compound
PGDB_C029725
6 activity records1 related patents
2D structure
N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCc7ccc(N8CCC(=O)NC8=O)cc7O6)CC5)CC4)nn3)CC2)cc1ClCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.52 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A000557 | PGDB_C029725 | PGDB_AS000481 | View |
| IC50 | - | = | 0.73 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001764 | PGDB_C029725 | PGDB_AS000195 | View |
| % Degradation | - | = | 50 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A001822 | PGDB_C029725 | PGDB_AS001838 | View |
| % Degradation | - | = | 61 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A003930 | PGDB_C029725 | PGDB_AS001354 | View |
| % Degradation | - | = | 40 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A006584 | PGDB_C029725 | PGDB_AS002389 | View |
| % Degradation | - | = | 43 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078536 | PGDB_C029725 | PGDB_AS002463 | View |