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Compound
PGDB_C029736
6 activity records1 related patents
2D structure
CCOC1(CN2CCC3(CC2)Oc2ccc(N4CCC(=O)NC4=O)cc2O3)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 70 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000017 | PGDB_C029736 | PGDB_AS001354 | View |
| % Degradation | - | = | 93 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000025 | PGDB_C029736 | PGDB_AS002389 | View |
| % Degradation | - | = | 69 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A006725 | PGDB_C029736 | PGDB_AS002463 | View |
| IC50 | - | = | 0.76 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078052 | PGDB_C029736 | PGDB_AS000195 | View |
| % Degradation | - | = | 93 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078064 | PGDB_C029736 | PGDB_AS001838 | View |
| IC50 | - | = | 0.00011 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A081199 | PGDB_C029736 | PGDB_AS000481 | View |